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Atividade antibacteriana in vitro de quatro espécies vegetais em diferentes gradua es alcoólicas In vitro antibacterial activity of four plant species at different alcoholic contents

Keywords: Fitoterapia , Escherichia coli , Staphylococcus aureus , Phytotherapy , Escherichia coli , Staphylococcus aureus

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Abstract:

Neste trabalho foi realizada a caracteriza o fitoquímica e avaliada a atividade antibacteriana in vitro dos extratos de Ageratum conyzoides L. (mentrasto), Gossypium hirsutum (algod o), Phyllanthus tenellus (quebra pedra), e Polygonum hydropiperoides (erva de bicho) frente à Staphylococcus aureus e Escherichia coli. Para a avalia o da atividade antibacteriana foi utilizado o método de difus o em ágar. Os testes foram realizados com o extrato nas gradua es alcoólicas de 0 a 100% (v/v), na propor o de 20% (m/v - massa/extrator). Os testes fitoquímicos constataram a presen a de a ucares redutores, compostos fenólicos, flavonoides, taninos, triterpenos, e esteróides nas quatro espécies. O crescimento das culturas de S. aureus foi inibido por todos os extratos, com exce o do extrato de Mentrasto. A maior atividade de inibi o foi observada pelo extrato de quebra pedra. Entretanto, nenhum dos extratos foi capaz de inibir o crescimento das cepas de E. coli. Os resultados s o promissores, visto que três das quatro plantas selecionadas demonstraram possuir substancias antibacterianas, o que motiva estudos subsequentes para o isolamento e identifica o dos princípios ativos responsáveis por essa atividade, com potencial de uso na indústria farmacêutica. In this study, phytochemical characterization was conducted and the in vitro antibacterial activity of extracts of Ageratum conyzoides L. (whiteweed), Gossypium hirsutum (cotton), Phyllanthus tenellus (shatterstone) and Polygonum hydropiperoides (swamp smartweed) was evaluated against Staphylococcus aureus and Escherichia coli. To assess the antibacterial activity, the agar diffusion method was used. Tests were performed with the extract at alcoholic contents from 0 to 100% (v/v), at 20% proportion (m/v - mass/extractor). Phytochemical tests indicated the presence of reducing sugars, phenolic compounds, flavonoids, tannins, triterpenes and steroids in all four species. The growth of S. aureus cultures was inhibited by all extracts, except for whiteweed extract. The highest inhibitory activity was observed for shatterstone. However, none of the extracts was capable of inhibiting the growth of E. coli strains. Results are promising since three of the four selected plants showed to have antibacterial substances, which stimulates further studies for the isolation and the identification of active principles responsible for this activity, with potential to be used in the pharmaceutical industry.

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